CM - Publications

2017

L. Halby, Y. Menon, E. Rilova, D. Pechalrieu, V. Masson, C. Faux, M.A. Bouhlel, M-H. David-Cordonnier, N. Novosad, Y. Aussagues, A. Samson, L. Lacroix, F. Ausseil, L. Fleury, D. Guianvarc'h, C. Ferroud, P. Arimondo. Rational design of bisubstrate-type analogs as inhibitors of DNA methyltransferases in cancer cells,  J. Med. Chem.2017, 60, 4665-4679

J. Jin, S. Guidi, Z. Abada, Z. Amara, M. Selva, M. W. George, M. Poliakoff, Continuous niobium phosphate catalysed Skraup reaction for quinoline synthesis from solketal, Green Chem. 2017, 19, 2439-2447

D. S. Lee, Z. Amara, C. A. Clark, Z. Xu, B. Kakimpa, H. P. Morvan, S. J. Pickering, M. Poliakoff, M. W. George, Continuous photo-oxidation in a vortex reactor: efficient operations using air drawn from the laboratory, Org. Process Res. Dev. 2017, 21, 1042-1050

Sylla-Iyarreta Veitía M., Siverio Mota D., Lerari V., Marín M., Giner R. M., Vicet Muro L., Rivero Guerra Y., Dumas F., Ferroud C., de Witte P. A. M., Crawford A. D., Arán V. J., Marrero Ponce Y., Fishing Anti-Inflammatories from Known Drugs: In Silico Repurposing, Design, Synthesis and Biological Evaluation of Bisacodyl Analogues, Curr. Top. Med. Chem., 2017, 17, 2866 – 2887,

Rayar A.-M., Lagarde N., Ferroud C., Zagury J.-F., Montes M., Sylla-Iyarreta Veitía M., Update on COX-2 Selective Inhibitors: Chemical Classification, Side Effects and their Use in Cancers and Neuronal Diseases, Curr. Top. Med. Chem., 2017, 17, 1-22.

M. Sylla-Iyarreta Veitía, F. Dumas, H. González-Díaz, Editorial: New Experimental and Computational Tools for Drug Discovery: From Chemistry to Biology. Curr. Top. Med. Chem.2017, 17, 2805 – 2806

2015-2016

Jorge, E.G. ; Rayar, A.M. ; Barigye, S.J. ; Rodriguez, M.E.J. ; Sylla-Iyarreta Veita, M. Development of an in Silico model of DPPH• free radical scavenging capacity: prediction of antioxidant activity of coumarin type compounds. Int. J. Mol. Sci., 2016, 17, 881 (Open access).

Sylla-Iyarreta Veitia M. and Ferroud C. New activation methods used in green chemistry for the synthesis of high value added molecules. Int. J. Energy Environ. Eng. 2015, 6, 37-46.

Renouard S., Corbin C., Colas C., Fidel T., Lopez T., Leclerc E.A., Hendrawati O., Falguières A., Doussot J., Ferroud C., Maunit B., Lainé E. and Hano C. Aerial part of Callitris species as a rich source of deoxypodophyllotoxin. Ind. Crops Prod., 2015, 63, 53-57.

Rayar A., Sylla-Iyarreta Veitia M., Ferroud C. An efficient and selective microwave-assisted Claisen-Schmidt reaction for the synthesis of functionalizedbenzalacetones. Springerplus, 2015, 4, 221 (Open access).

Görmen M., Sylla-Iyarreta Veitia M., Trigui F., El Arbi M., Ferroud C. Ferrocenyl derivatives of bisacodyl: synthesis and antimicrobial activity. J. Organomet. Chem. 2015, 794, 274-281.

2013-2014

F. Dioury, A. Duprat, G. Dreyfus, C. Ferroud, J. Cossy, QSPR Prediction of the Stability Constants of Gadolinium(III) Complexes for MRI, J. Chem. Inf. Model. 2014, 54, 2718–2731

G. Bort, S. Catoen, H. Borderies, A. Kebsi, S. Ballet, G. Louin, M. Port, C. Ferroud, Gadolinium-based contrast agents targeted to amyloid aggregates for the early diagnosis of Alzheimer's disease by MRI, Eur. J. Med. Chem. 2014, 87, 843-861.

M. Wagner, Y. Contie, C. Ferroud, G. Revial. Enantioselective Aldol Reactions and Michael Additions Using Proline Derivatives as Organocatalysts IJOC, 2014, 4, 55-67 (Open access).

O. Fliniaux, C. Corbin, A. Ramsay, S. Renouard, V. Beejmohun, J. Doussot, A. Falguière, C. Ferroud, F. Lamblin, E. Lainé, A. Rosche, E. Grand, F. Mesnard and C. Hano, Microwave-Assisted Extraction of Herbacetin Diglucoside from Flax (Linum usitatissimum L.) Seed Cakes and Its Quantification using an RP-HPLC-UV System. Molecules, 2014, 19, 3025-3037 (Open access)

G. Bort, M. Sylla-Iyarreta Veitía, C. Ferroud, Straightforward synthesis of PET tracer precursors used for the early diagnosis of Alzheimer's disease through Suzuki-Miyaura cross-coupling reactions. Tetrahedron, 2013, 69, 7345-7353

C. Ricco. 1,3-Diiodo-5,5-dimethylhydantoin. Synlett, 2013, 24, 2173–2174 (Spotlight)

2011-2012

C. Ferroud; G. Revial; R. Morfin. Chemical and biochemical approaches to the production of 7-hydroxylated C19-steroids. Horm. Mol. Biol. Clin. Invest., 2012, 10, 293-300.

I. Idri, J-L. Havet, J. M. Garcia Fernandez, C. Ferroud, C. Porte; Microwave-assisted synthesis of prebiotic di-D-fructose dianhydride-enriched caramels. Food Chem., 2012, 134, 1527–1532

M. .Biasutti, N. Dufour, C. Ferroud, W. Dab, L. Temime; Cost-Effectiveness of Magnetic Resonance Imaging with a New Contrast Agent for the Early Diagnosis of Alzheimer's Disease, PLoS ONE, 2012, 7, e35559 (Open access)

K. Fidaly, C. Ceballos, A. Falguières, M. Sylla-Iyarreta Veitia, A. Guy, C. Ferroud. Visible light photoredox organocatalysis: a fully metal-free direct asymmetric α-alkylation of aldehydes. Green Chem., 2012, 14, 1293-1297.

L. Halby, C. Sénamaud-Beaufort, S. Ajjan, A. Ceccaldi, T. Drujon, A. Rajavelu, C. Champion, R. Jurkowska, O. Lequin, W. G. Nelson, A. Jeltsch, A. Guy, D. Guianvarc’h, C. Ferroud and P. B. Arimondo; Rapid synthesis of new DNMT inhibitors derivatives of procainamide. ChemBioChem., 2012, 13, 157-165

Guianvarc’h, D.; Arimondo, P.; Senamaud-Beaufort, C.; Grellier, P.; Halby, L.; Ferroud, C. Substituted amino - benzoic acid derivatives as inhibitors of DNA methyltransferases. (20 septembre 2011), PCT/EP2011/066305 (WO2012/038417)

C. Ricco, G. Revial, C. Ferroud, O. Hennebert, R. Morfin; Synthesis of a 19-(O-carboxymethyl)oxime hapten of 7beta-hydroxy-epiandrosterone. Horm. Mol. Biol. Clin. Invest., 2011, 7, 295-301.

M. D. Altmtop, Z. A. Kaplancikli, G. Turan-Zitouni, A. Ozdemir, F. Demirci, G. Iscan, G. Revial. Synthesis of some novel triazole derivatives and investigation of their antimicrobial activities. Synth. Commun., 2011, 41, 2234-2250.

M. Sylla-Iyarreta Veitía, M. Joudat, M. Wagner, A. Falguières, A. Guy, C. Ferroud, Ready available chiral azapyridinomacrocycles N-oxides; first results as Lewis base catalysts in asymmetric allylation of p-nitrobenzaldehyde. Heterocycles, 2011, 83, 2011-2039.

S. Renouard, T. Lopez, O. Hendrawati, J. Doussot, P.Dupré, A. Falguières, C. Ferroud, D. Hagège, F. Lamblin, E. Lainé and C. Hano. Podophyllotoxin and deoxypodophyllotoxin in Juniperus bermudiana and 12 other Juniperus species – optimization of extraction, method validationand quantification. J. Agric. Food Chem., 2011, 59, 8101-8107.

M. Petit, G. Bort, B-T. Doan, C. Sicard, D. Ogden, D. Scherman, C. Ferroud, P. I. Dalko, X-ray photolysis to release ligands from caged Reagents by an intramolecular antenna sensitive to magnetic resonance imaging. Angew. Chem., 2011, 50, 9708-9711.

L. Rakotozafy, A. Falguières, M. Sidibe, C. Ferroud, J. Potus, J. Nicolas,  Effets de l’addition de peroxyde d’hydrogène sur l’oxydation de deux phénols (tyrosine, acide férulique) et d’un thiol (glutathion) présents dans un extrait aqueux de farine; analyse par CLHP-DAD et CLHP-SM. Industries des céréales, 2011, 174, 20-24.

C. Ricco, G. Revial, C. Ferroud, O; Hennebert, R. Morfin; Synthesis of 7 ß-hydroxy-epiandrosterone. Steroids, 2011, 76, 28-30.

2009-2010

L. Rakotozafy, M. Sidibe, A. Falguières, V. Lemaître, C. Ferroud, J. Potus, J. Nicolas ; Oxydation de la tyrosine par la peroxydase du blé en présence de cystéine, glutathion et d’acides cinnamiques. Industries des céréales, 2010, 169, 10-16

A. Ozdemir, G. Turan-Zitouni, Z.A. Kaplancikli, G. Revial, F. Demirci, G. Iscan Preparation of some pyrazoline derivatives and evaluation of their antifungal activities. J. Enzyme Inh. Med. Chem. , 2010, 25, 565-571.

Olivier Hennebert, Matthieu Montes, Alain Favre-Reguillon, Henry Chermette, Clotilde Ferroud, Robert Morfin ; Epimerase activity of the human 11-hydroxysteroid dehydrogenase type 1 on 7-hydroxylated C19-steroids; J. Steroid Biochem. Mol. Biol;, 2009, 114, 57-63

Xie, L.-L.; Favre-Reguillon, A.; Wang, X.-X.; Fu, X.; Vrinat, M.; Lemaire, M.; Selective Extraction of Neutral Nitrogen-Containing Compounds from Straight-Run Diesel Feed Using Polymer-Supported Ionic Liquid MoietiesInd. Eng. Chem. Res., 2009, 48, 3973-3977

Synthesis of an hexadentate tricyclic tetraazadiacetic ligand as precursor for MRI contrast enhancement agent; F. Dioury, C. Ferroud, A. Guy, and M. Port, Tetrahedron, 2009, 65, 7573-7579

Synthesis of novel N-protected β3-amino nitriles: study of their hydrolysis involving a nitrilase-catalysed step; M. Sylla-Iyarreta Veitia, P-L. Brun, P. Jorda, A. Falguières et C. Ferroud, Tetrahedron : Asymmetry, 2009, 20, 2077-2089

Synthesis, structural analysis and anticonvulsant activity of a ternary Cu(II) mononuclear complex containing 1,10-phenanthroline and the leading antiepileptic drug valproic acid. M Sylla-Iyarreta Veitia, F. Dumas, G. Morgant, J. R. J. Sorenson,Y. Frapart, A. Tomas, Biochimie, 2009, 91, 1286-1293

Synthesis Characterization and biological activities of metal-base complexes containning the leading drug valproic acid. M. Sylla-Iyarreta Veita, F. Dumas, G. Morgant, Brevet no PCT/FR2009/051077 (8 juin 2009)

2007-2008

Synthesis of a novel amphiphilic GdPCTA-[12] derivative as a potantial micellar MRI contrast agent, Clotilde Ferroud, Hélène Borderies, Elizabeth Lasri, Alain Guy, Marc Port Tetrahedron Lett., 2008, 49, 5972-5975

Microwaves assisted N-acetamides synthesis by amidation or aminolysis, Clotilde Ferroud, Ung Stéphane, Godart Marie, Borderies Hélène and Guy Alain, Tetrahedron Lett., 2008, 49, 3004-3008

New triazole and triazolothiadiazine derivatives as possible antimicrobial agents
Z.A. Kaplancikli, G. Turan-Zitouni, A.Özdemir, G. Revial European Journal of Medicinal Chemistry, 2008, 43, 155-159

Synthesis and anticandidal activity of some imidazopyridine derivatives. Z.A. Kaplancikli, G. Turan-Zitouni, A.Özdemir, G. Revial. Journal of Enzyme Inhibition and Medicinal Chemistry, 2008, 23(6), 866-870

Selective extraction of neutral nitrogen compounds found in diesel feed by 1-butyl-3-methyl-imidazolium chloride; Xie, L.-L.; Favre-Reguillon, A.; Wang, X.-X.; Fu, X.; Pellet-Rostaing, S.; Toussaint, G.; Geantet, C.; Vrinat, M.; Lemaire, M. Green Chemistry, 2008, 10, 524-531

Selective Extraction and Identification of Neutral Nitrogen Compounds Contained in Straight-Run Diesel Feed Using Chloride Based Ionic Liquid; Xie, L.-L.; Favre-Reguillon, A.; Pellet-Rostaing, S.; Wang, X.-X.; Fu, X.; Estager, J.; Vrinat, M.; Lemaire, M.; Ind. Eng. Chem. Res., 2008, 47, 8801-8807

Sequestering agents for uranyl chelation: new calixarene ligands; Leydier, A.; Lecercle, D.; Pellet-Rostaing, S.; Favre-Reguillon, A.; Taran, F.; Lemaire, M.; Tetrahedron, 2008, 64, 11319-11324

Deep desulfurization of diesel feedstock by selective adsorption of refractory sulfur compounds; Favre-Reguillon, A.; Sevignon, M.; Rocault, M.; Schulz, E.; Lemaire, M.; Ind. Eng. Chem. Res., 2008, 47, 9617-9622

Removal of N-compounds from diesel fuel by using chloridized imidazole based ionic liquids; Xie, L.-L.; Chen, X.; Wang, X.-X.; Fu, X.-Z.; Favre-Reguillon, A.; Pellet-Rostaing, S.; Lemaire, M.; Wuji Huaxue Xuebao, 2008, 24, 919-925

Synthesis of original capping calixarenes with DTPA fragment; Lin, Y.; Leydier, A.; Metay, E.; Favre-Reguillon, A.; Bouchu, D.; Pellet-Rostaing, S.; Lemaire, M.; Journal of Inclusion Phenomena and Macrocyclic Chemistry, 2008, 61, 187-193

Radiation chemistry of cis-syn-cis dicyclohexano-18-crown-6 (DCH18C6): Acidity and uranyl nitrate dependence; Draye, M.; Favre-Reguillon, A.; Faure, R.; Lemaire, M.; Radiat. Phys. Chem., 2008, 77, 581-584

Sequestering agent for uranyl chelation: a new family of CAMS ligands; Leydier, A.; Lecercle, D.; Pellet-Rostaing, S.; Favre-Reguillon, A.; Taran, F.; Lemaire, M.; Tetrahedron, 2008, 64, 6662-6669

Selective removal of dissolved uranium in drinking water by nanofiltration; Favre-Reguillon, A.; Lebuzit, G.; Murat, D.; Foos, J.; Mansour, C.; Draye, M.; Water Res., 2008, 42, 1160-1166

Synthesis of a tricyclic tetraazatriacetic ligand for gadolinium (III) as potential contrast agent for MRI. F.Dioury, S. Sambou, E. Guéné, M. Sabatou, C. Ferroud, A. Guy and M. Port; Tetrahedron, 2007, 63, 204-214

7alpha- and 7beta-Hydroxy-epiandrosterone as substrates and inhibitors for the human 11-hydroxysteroid dehydrogenase type 1. O. Hennebert, C. Pernelle, C. Ferroud and R. Morfin; J. Steroid Biochem. Mol. Biol., 2007, 105, 159-165

2004-2006

Impact of rigidification on relaxometric properties of a tricyclic-tetraazatriacetic gadolinium chelate ; M. Port, I. Raynal, L. Vander Elst, R. N. Muller, F. Dioury, C. Ferroud, A. Guy, Contrast Med. Mol. Imaging, 2006, 1, 121-127

Quatre expériences de formation à distance dans le pôle Sciences et Techniques Industrielles du Cnam Paris. M. Debacq, M. Clausse, V. Dalmeyda, J-P. Domblides, C. Ferroud, G. Villoutrex ; Proceeding, Technologies Information Communication Enseignement, TICE 2006, Toulouse, 25-27 octobre 2006

Synthesis of a new tricyclic tetraazatriacetic acid as ligand for gadolinium (III); F. Dioury, E. Guéné, A. Di Scala-Roulleau, C. Ferroud, A. Guy et M. Port, Tetrahedron Lett., 2005, Vol 46(4), 611-613

Chemoselective ultrasonically activated reduction of substituted nitrobenzenes to corresponding N-hydroxylamines; S. Ung, A. Falguières, A. Guy and C. Ferroud, Tetrahedron Lett., 2005, 46, 5913-5917

Regioselectively N-Functionalized 14-Membered Azapyridinomacrocycles Bearing Trialkylcarboxylic Acid Side Chains as Ligands for Lanthanide Ions, F. Dioury, I. Sylvestre, J-M. Siaugue, V. Wintgens, C. Ferroud, A. Favre-Réguillon, J. Foos, and A. Guy, Eur. J. Org. Chem. 2004, 21, 4424-4436.

C-ACTI (Communication avec actes, colloque international)

Moreau, G. ; Fourati, N. ; Zerrouki, C. ; Mouhsine, H. ; Montes, M. ; Port, M. ; Sylla-Iyarreta Veitia, M. ; Zagury, J.F. ; Yaakoubi, N. 2016. Surface acoustic wave biosensors for the quantification of TNFα/SPD304 interaction. Congrès Eurosensors 2016, Budapest, septembre 2016.

Rayar A., Goya Jorge E., Jones Barigye S., Jorge Rodriguez M., Ferroud C. and Sylla-Iyarreta Veitia M. 2015. Microwave assisted synthesis of Benzalacetones and study of their potential antioxidant activity using artificial neural networks method. In  Proceedings of the MOL2NET, 5-12 december, Sciforum Electronic Conference Series, vol. 1, b028.

Görmen M., Sylla-Iyarreta Veitia M., Trigui F., El Arbi M., Ferroud C. 2015. Conception, synthesis, characterization and antimicrobial evaluation of new ferrocene-based derivatives inspired by the bisacodyl lead structure. In  Proceedings of the MOL2NET, 5-12 december, Sciforum Electronic Conference Series, vol. 1, b021.

Goya Jorge E., Rayar A., Jones Barigye S., Jorge Rodriguez M. and Sylla-Iyarreta Veitia M. 2015. Free radical scavenging activity of coumarin derivatives. In silico and in vitro approach. 2015. In  Proceedings of the MOL2NET, 5-12 december, Sciforum Electronic Conference Series, vol. 1, b024.

Sylla Iyarreta Veitia M., Rampal C. and Ferroud C. 2015. Regioselective Friedel-Crafts hydroalkylation using friendly conditions: application to the synthesis of unsymmetrical triarylmethanes. In Proceedings of the MOL2NET, 5-12 december, Sciforum Electronic Conference Series, vol. 1, a006.

Sylla Iyarreta Veitia M. ; Siverio Mota D. ; Lerari V. ; Vicet Muro L. ; Rivero-Guera M. ; Marin M. ; Giner R.M. ; Ferroud C. ; De Witte P. ; Crawford A.D. ; Aran V.J. ; Marrero Ponce C.Y. 2014. In silico repurposing, design, synthesis and biological evaluation of new analogues of bisacodyl as potential anti-inflammatory agents. XXIII International Symposium on medicinal chemistry (Lisbonne, Portugal) 7-11 septembre.

Sylla-Iyarreta Veitia M. ; Ferroud C. 2014. La chimie verte au Cnam : catalyse enzymatique et activation physicochimique par microonde pour la synthèse de molecules à haute valeur ajoutée. Cofret’14 colloque francophone en énergie, environnement, économie et thermodynamique (Paris, France) 23-25 avril.

Towards big data in QSAR/QSPR, A. Duprat, F. Dioury, J.-L. Ploix, G.Dreyfus, acte de congrès du 24th IEEE International Workshop on Machine Learning for Signal Processing (MLSP2014), 21-24 septembre 2014, Reims, France, publication acceptée.

C-ACTN (Communication avec actes, colloque national)

Yong-Sang, J. ; Dioury, F. ; Jestin, E. ; Ferroud, C. ; Meilhac, O. 2016. Nouvel outil de diagnostic en imagerie TEP de l’athérothrombose et de l’ischémie cérébrale. Ma thèse en 180 secondes, doctoriales de l’ED Sciences Technologies Santé (ED 542), Université de La Réunion, Saint Gilles les Bains, 8 avril 2016.

Rayar, A. ; Lagarde, N. ; Ferroud, C. ; Zagury, J.F. ; Sylla-Iyarreta Veitia, M. ; Montes, M. 2016. In silico drug design and medicinal chemistry: development of new unusual structures targeting the Cyclooxygenase-2. 23ème journées jeunes chercheurs de la société de chimie thérapeutique, Lille, 15-17 février 2016.

Rayar, A. ; Lagarde, N. ; Ferroud, C. ; Zagury, J.F. ; Sylla-Iyarreta Veitia, M. ; Montes, M. 2016. Development of original selective cyclooxygenase-2 inhibitors: pharmacophores design and synthesis. 20ème journée de chimie organique et chimie organique biologique de la montagne sainte Geneviève, Paris, juin 2016.

La chimie verte au Cnam : catalyse enzymatique et activation physicochimique par micro-ondes pour la synthèse de molécules à haute valeur ajoutée. M. Sylla-Iyarreta Veitía et C. Ferroud. COlloque FRancophone en Energie, Environnement, Economie et Thermodynamique (COFRET'14), Paris, Cnam du 23 au 25 avril 2014, Volume de 1154 pages, ISSN 2269-1901